API reference
Fesoterodine fumarate
- CAS number
- 286930-03-8
- Molecular formula
- C30H41NO7
- Molecular weight
- 527.6 g/mol
About this molecule
Fesoterodine Fumarate is the fumarate salt form of fesoterodine, a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties. Fesoterodine is rapidly hydrolyzed in vivo into its active metabolite 5-hydroxy methyl tolterodine, which binds and inhibits muscarinic receptors on the bladder detrusor muscle, thereby preventing bladder contractions or spasms caused by acetylcholine. This results in the relaxation of bladder smooth muscle and greater bladder capacity, in addition to a reduction in involuntary muscle contractions and involuntary loss of urine. The active metabolite does not interact with alpha-adrenergic, serotonergic, histaminergic and excitatory amino acid receptors and is eliminated via renal excretion.
Source: NCI Thesaurus (NCIt), via PubChem.
Identifiers
- IUPAC name
- (E)-but-2-enedioic acid;[2-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-(hydroxymethyl)phenyl] 2-methylpropanoate
- InChIKey
- MWHXMIASLKXGBU-RNCYCKTQSA-N
- SMILES
- CC(C)C(=O)OC1=C(C=C(C=C1)CO)[C@H](CCN(C(C)C)C(C)C)C2=CC=CC=C2.C(=C/C(=O)O)\C(=O)O
- PubChem CID
- 9849808
Also known as
Fesoterodine fumarate · Toviaz · SPM 907 · SPM-907 · (R)-Fesoterodine fumarate · Fesoterodine (fumarate) · C30H41NO7 · Toviaz (TN)
Chemical data on this page is drawn from PubChem (National Library of Medicine) and is provided for identification only. Hanpars does not hold stock of every substance listed; availability, grade, documentation and regulatory status are confirmed per enquiry.
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