API reference
Remimazolam besylate
- CAS number
- 1001415-66-2
- Molecular formula
- C27H25BrN4O5S
- Molecular weight
- 597.5 g/mol
About this molecule
Remimazolam Besylate is the besylate ester form of remimazolam, a short-acting benzodiazepine derivative that is structurally related to midazolam, with sedative-hypnotic activity. Upon administration, remimazolam targets and binds to a specific site on the gamma-aminobutyric acid (GABA)-A-chloride ionophore receptor complex located on the neuronal membrane. Binding causes an allosteric modification of the receptor thereby enhancing the affinity of GABA to the receptor leading to an increase in the frequency of chloride-channel opening events, which leads to an increase in chloride ion conductance, neuronal hyperpolarization, inhibition of the action potential, and a decrease in neuronal excitability.
Source: NCI Thesaurus (NCIt), via PubChem.
Identifiers
- IUPAC name
- benzenesulfonic acid;methyl 3-[(4S)-8-bromo-1-methyl-6-pyridin-2-yl-4H-imidazo[1,2-a][1,4]benzodiazepin-4-yl]propanoate
- InChIKey
- QMTKNJZIWGTNTE-LMOVPXPDSA-N
- SMILES
- CC1=CN=C2N1C3=C(C=C(C=C3)Br)C(=N[C@H]2CCC(=O)OC)C4=CC=CC=N4.C1=CC=C(C=C1)S(=O)(=O)O
- PubChem CID
- 23658607
Also known as
Remimazolam Benzenesulfonate · Remimazolam Besylate · BIPRAZINE PF · Byfavo · SP148.5 · anerem · Remimazolam besilate · Remimazolam (benzenesulfonate)
Chemical data on this page is drawn from PubChem (National Library of Medicine) and is provided for identification only. Hanpars does not hold stock of every substance listed; availability, grade, documentation and regulatory status are confirmed per enquiry.
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